| 编号 | 中文名 | English Name | 分子式 | CAS.NO | 备注 |
| 1 | 托吡司特 | Topiroxostat | C13H8N6 | 577778-58-6 | Y20230000309 |
| 2 | 达普司他 | Daprodustat | C19H27N3O6 | 960539-70-2 | Y20230000043 |
| 3 | 左西孟旦 | Levosimendan | C14H12N6O | 141505-33-1 | Y20220001079 |
| 4 | 富马酸伏诺拉生 | Vonoprazan Fumarate | C21H20FN3O6S | 260141-27-2 | Y20220000944 |
| 5 | 达可替尼 | Dacomitinib | 1110813-31-4 | C24H25ClFN5O2 | Y20220000939 |
| 6 | 美阿沙坦钾 | Azilsartan Medoxomil Potassium | C30H23KN4O8 | 863031-24-7 | Y20220000851 |
| 7 | 艾拉戈克钠 | Elagolix Sodium | C32H29F5N3NaO5 | 832720-36-2 | Y20220000614 |
| 8 | 利格列汀 | Linagliptin | C25H28N8O2 | 668270-12-0 | Y20220000539 |
| 9 | 碳酸镧 | Lanthanum Carbonate | C3La2O9 | 587-26-8 | Y20220000402 |
| 10 | 氢溴酸伏硫西汀 | Vortioxetine Hydrobromide | C18H23BrN2S | 960203-27-4 | Y20220000220 |
| 11 | 恩格列净 | Empagliflozin | C23H27ClO7 | 864070-44-0 | Y20210001250 |
| 12 | 阿普米司特 | Apremilast | C22H24N2O7S | 608141-41-9 | Y20200001491 |
| 13 | 赛洛多辛 | Silodosin | C25H32F3N3O4 | 160970-54-7 | Y20210000365 |
| 14 | 盐酸培唑帕尼 | Pazopanib Hydrochloride | C21H24ClN7O2S | 635702-64-6 | Y20210000469 |
| 15 | 盐酸普拉格雷 | Prasugrel hydrochloride | C20H21ClFNO3S | 389574-19-0 | Y20210000621 |
| 16 | 甲磺酸仑伐替尼 | Lenvatinib Mesilate | C22H23ClN4O7S | 57890-39-2 | Y20210000659 |
| 17 | 甲磺酸萘莫司他 | Nafamostat mesilate | C21H25N5O8S2 | 82956-11-4 | Y20200001018 |
| 18 | 苹果酸舒尼替尼 | Sunitinib Malate | C26H33FN4O7 | 341031-54-7 | Y20200000781 |
| 19 | 盐酸左布比卡因 | Levobupivacaine Hydrochloride | C18H29ClN2O | 27262-48-2 | Y20190021493 |
| 20 | 磷酸西格列汀 | Sitagliptin Phosphate | C16H20F6N5O6P | 654671-77-9 | Y20190021505 |
| 21 | 盐酸奥普力农 | Olprinone HCl | C14H11ClN4O | 119615-63-3 | Y20200000291 |
| 22 | 酒石酸伐尼克兰 | Varenicline Tartrate | C17H19N3O6 | 375815-87-5 | Y20190021278 |
| 23 | 富马酸丙酚替诺福韦 | Tenofovir Alafenamide Fumarate | C46H62N12O14P2 | 1392275-56-7 | Y20190021425 |
| 24 | 普拉洛芬 | Pranoprofen | C15H13NO3 | 52549-17-4 | Y20190021277 |
| 25 | 拉考沙胺 | Lacosamide | C13H18N2O3 | 175481-36-4 | Y20190001000 |
| 26 | 帕瑞昔布钠 | Parecoxib | C19H18N2O4S | 198470-84-7 | Y20190000999 |
| 27 | 米拉贝隆 | Mirabegron | C21H24N4O2S | 223673-61-8 | Y20180001417 |
| 28 | 盐酸达泊西汀 | Dapoxetine Hydrochloride | C21H24ClNO | 129938-20-1 | Y20180001416 |
| 29 | 盐酸伐地那非 | Vardenafil Hydrochloride | C23H33ClN6O4S | 224785-91-5 | Y20180001528 |
| 30 | 甲苯磺酸索拉非尼 | Sorafenib Tosylate | C28H24ClF3N4O6S | 475207-59-1 | Y20180000277 |
| 31 | 琥珀酸普芦卡必利 | Prucalopride Succinate | C22H32ClN3O7 | 179474-85-2 | Y20180000320 |
| 32 | 非布司他 | Febuxostat | C16H16N2O3S | 144060-53-7 | Y20200000278 |
| 33 | 盐酸西那卡塞 | Cinacalcet Hydrochloride | C22H23ClF3N | 364782-34-3 | Y20180000458 |
| 34 | 塞来昔布 | Celebrex | C17H14F3N3O2S | 169590-42-5 | Y20180000610 |
| 35 | 阿哌沙班 | Apixaban | C25H25N5O4 | 503612-47-3 | Y20180000609 |
| 36 | 地氯雷他定 | Desloratadine | C19H19ClN2 | 100643-71-8 | Y20180000860 |
| 37 | 维格列汀 | Vildagliptin | C17H25N3O2 | 274901-16-5 | Y20180000901 |
| 38 | 盐酸厄洛替尼 | Erlotinib Hydrochloride | C22H24ClN3O4 | 183319-69-9 | Y20180001037 |
| 39 | 依折麦布 | Ezetimibe | C24H21F2NO3 | 163222-33-1 | Y20180001036 |
| 40 | 盐酸托莫西汀 | Atomoxetine Hydrochloride | C17H22ClNO | 82248-59-7 | Y20180001108 |
| 41 | 吉非替尼 | Gefitinib | C22H24ClFN4O3 | 184475-35-2 | Y20180001109 |
| 42 | 依托考昔 | Etoricoxib | C18H15ClN2O2S | 202409-33-4 | Y20180001167 |
| 43 | 瑞舒伐他汀钙 | RosuvastatinCalcium | C44H54CaF2N6O12S2 | 147098-20-2 | Y20170001976 |